[1 ] Houghten R A , Perspectives in Drug Discoveryand Design, 1995, 2 (2).
[2 ] Weintraub H, Science, 1995, 267, 1609.
[3 ] Terrett N K, Gardner M , Gordon D W , Kobylecki R J , Steele J , Tetrahetron, 1995, 51 (30) , 8135~8173.
[4 ] Nielsen J , Chemistry & Industry , 1994, 902~ 905.
[5 ] Brown K D, Genetic Engineering News, 1992, 12 (19) , 1.
[6 ] Jung G, Beck-Sickinger A G, Angew. Chem. Int. Ed. Engl. , 1992, 31 (4) , 367~ 486.
[7 ] Jacobs J W , Trendsin Biotechnology , 1994, 12 (1) , 19~ 26.
[8 ] Janda K D, Proc. Natl. Acad. Sci. USA , 1994, 91, 10779~ 10785.
[9 ] Gallop M A , Barrett R W , Dower W J , Fordor S P A , Gordon E M , J. Med. Chem. , 1994, 37 (9) ,1233~ 1251.
[10 ] Gordon E M , Barrett R W , Dower W J , Fordor S P A , Gallop M A , J. Med. Chem. , 1994, 37(10) , 1385~ 1400.
[11 ] Vries D J , Hall M R, Drug Development Research, 1994, 33, 161~ 173.
[12 ] Furka A , Drug Development Research, 1994, 33, 90~ 97.
[13 ] Ellington A D, Drug Development Research, 1994, 33 (2) , 102~ 115.
[14 ] Clackson T , Well J A , Trends in Biotechnology , 1994, 12 (5) , 173~ 184.
[15 ] Houghten R A , Technical Focus, 1993, 9 (7) , 235~ 239.
[16 ] Pavia M R, Sawyer T K, Moos W H, Bioorganic &Medicinal Chemistry Letters, 1993, 3 (3) , 387~396.
[17 ] 刘刚, 中国药物化学杂志, 1995, 5 (4) , 303~ 310.
[18 ] 刘刚, 中国药物化学杂志, 1996, 6 (1) , 73~ 78.
[19 ] Lebl M , Krchnak V , Sepetov N F, Seligmann B, Strop P, Felder S, Lam K S, Biopolymers (Peptide Science) , 1995, 37, 177~ 198.
[20 ] Lam K S, Lebl M , Methods: A Companion to Methods in Enzymology , 1994, 6, 372~ 380.
[21 ] Martin E J , Blaney J M , Siani M A et al. , J. Med. Chem. , 1995, 38, 1431~ 1436.
[22 ] Zuckmann R N , Martin E J , Spellmeyer D C et al. , J. Med. Chem. , 1994, 37, 2678.
[23 ] Eichler J , Lucka A W , Houghten R A , Peptide Research, 1994, 7, 300.
[24 ] Madden D, Krchnak V , Lebl M , Perspectivesin Drug Discoveryand Design, 1995, 2, 269~ 285.
[25 ] Stankova M , Issakova O S, Drug Dev. Res. , 1994, 33, 146.
[26 ] Geysen H M , Meloen R H, Barteling S J , Proc. Natl. Acad. Sci. USA , 1984, 81, 3998.
[27 ] Houghten R A , Proc. Natl. Acad. Sci. USA , 1985, 82, 5131.
[28 ] Fodor S P A , Read J L , Pirrung M C, Stryer L , Lu A T , Solas D, Science, 1991, 251, 767.
[29 ] Berg R H, Almdal K, Pedersen W B, Peptides, Chemistry Structure and Biology , Proc. 11th Am.Pept. Symp (eds. River J E, Marshall G R) , Escom , Leiden, 1990, 1036.
[30 ] Berg R H, Almdal K, Pedersen W B, Peptides, 1990: Proc. 21st Eur. Pept. Symp. (eds. Giralt E,Andreu D) , Escom , Leiden, 1991, 149.
[31 ] Frank R, Doring R, Tetrahedron, 1988, 44, 6031.
[32 ] Lam K S, Salmon S E, Hersh E M , Hruby V J , Kazmierski W M , Knapp R J , Nature, 1991, 354,82~ 84.
[33 ] Furka A , Sebestyen F, Dibo G, Int. J. Peptide Protein Res. , 1991, 37, 487~ 493.
[34 ] Lebl M , Krchnak V , Sepetov N F, Seligmann B, Strop P, Felder S, Lam K S, Biopolymers,1995, 37, 177~ 198.
[35 ] Houghten R A , Pinilla C, Blondelle S E, Appel J R, Dooley C T , Cuervo J H, Nature, 1991, 354,84.
[36 ] Blondelle S, The 2nd European Conferenceon High Throughput Screening and on Exploiting Molecular Diversity , May 17~ 20, 1995, Abstract.
[37 ] Cwirla S E, Peters E A , Barrett P R W , Dower W J , Proc. Natl. Acad. Sci. USA , 1990, 87, 6378~ 6382.
[38 ] Scott J K, Smith G P, Science, 1990, 249, 386~ 390.
[39 ] Barrett R W , Cwirla S E, Ackerman M S, Olson A M , Peters E A , Dower W J , Analytical Biochemistry , 1992, 204, 357~ 364.
[40 ] Felici F, J. Mol. Biol. , 1991, 222, 301~ 310.
[41 ] Hoogenboom H R, Griffiths A , Johnson K S, Chiswell D J , Hudson P, Winter G, Nucleic Acids Research, 1991, 19 (15) , 4133~ 4137.
[42 ] Marks J D, Hoogenboom H R, Bonnert T P, McCafferty J , Griffiths A D, Winter G, J. Mol. Biol. ,1991, 222, 581~ 597.
[43 ] Greenwood J , Willis A E, Perham R N , J. Mol. Biol. , 1991, 220, 821~ 827.
[44 ] Fong S, Doyle L V , Devlin J J , Doyle M V , Drug Development Research, 1994, 33, 64~ 70.
[45 ] KangA S, Barbas C F, Janda K D, Benkovic S J , Lerner R A , Proc. Natl. Acad. Sci. USA , 1991,88, 4363~ 4366.
[46 ] Koivunen E, Wang B C, Ruoslahti E, Bio/Technology , 1995, 265~ 270.
[47 ] Hagihara M , Anthony N J , Stout T J , Clardy J , Schreiber S L , J. Am. Chem. Soc. , 1992, 114, 6568~ 6570.
[48 ] Egholm M , Buchardt O , Nielsen P E, Perg R H, J. Am. Chem. Soc. , 1992, 114, 1895~ 1897.
[49 ] Simon R J , Kania R S, Zuckermann R N , Huebner V D, Jewell D A , Banville S, Ng S, Wang L ,Rosenberg S, Marlowe C K, SpellmeyerD C, Tan R, FrankelA D, SantiD V , Cohen F E, Bartlett P A , Proc. Natl. Acad. Sci. USA , 1992, 89, 9367~ 9371.
[50 ] Smith A B, Keenan T P, Holcomb R C, Sprengeler P, GuzmanM C, Wood J L , Carroll P J ,Hirschmann R, J. Am. Chem. Soc. , 1992, 114, 10672~ 10674.
[51 ] Cho C Y, Moran E J , Cherry S R, Stephans J C, Fordor S P A , Adams C L , Sundaram A , Jacobs J W , Schultz P G, Science, 1993, 261, 1303~ 1305.
[52 ] Zuckermann R N , Kerr J M , Kent S B H, Moos W H, J. Am. Chem. Soc. , 1992, 114, 10646~10647.
[53 ] Miller S M , Simon R J , Ng S, Zuckermann R N , Kerr J M , Moos W H, Bioorganic &Medicinal Chemistry Letters, 1994, 4 (22) , 2657~ 2662.
[54 ] HowellD C, Howson W , Rees D C, Drug Designand Discovery , 1994, 12, 63~ 75.
[55 ] Danishefsky S J , McClure K F, Randolph J T , Ruggeri R B, Science, 1993, 260, 1307~ 1309.
[56 ] Douglas S P, Whitfield D M , Krepinsky J J , J. Am. Chem. Soc. , 1991, 113, 5095~ 5097.
[57 ] SchusterM , Wang P, Paulson J C, Wong C H, J. Am. Chem. Soc. , 1994, 116, 1135~ 1136.
[58 ] Vetter D, Gallop M A , Bioconjugate Chemistry , 1995, 6, 316~ 318.
[59 ] Vetter D, Tate EM , Gallop M A , Bioconjugate Chemistry , 1995, 6, 319~ 322.
[60 ] Brenner S, Lerner R A , Proc. Natl. Acad. Sci. USA , 1992, 89, 5381~ 5383.
[61 ] Needels M C, Brenner S, Janda K D, J. Am. Chem. Soc. , 1993, 115, 9812~ 9813.
[62 ] Needels M C, Jones D G, Tate E H, Heinkel G L , Kochersperger L M , Dower W J , Barrett R W Gallop M A , Proc. Natl. Acad. Sci. USA , 1993, 90, 10700~ 10704.
[63 ] Ohlmeyer M H J , Swanson R N , Dillard L W , Reader J C, Asouline G, Kobayashi R, Wigler M ,Still W C,ibid. , 1993, 90, 10922~ 10926.
[64 ] Borchard A , Still W C, J. Am. Chem. Soc. , 1994, 116, 373~ 374.
[65 ] Kerr J M , Banville S C, Zuckermann R N , J. Am. Chem. Soc. , 1993, 115, 2529~ 2531.
[66 ] Nicolaou K C, Xiao X Y, Parandoosh Z et al. , Angew. Chem. Int. Ed. Engl. , 1995, 34 (20) , 2289~ 2291.
[67 ] Siani M A , Weininger D, Blaney J M , J. Chem. Inf . Comput. Sci. , 1994, 34, 588~ 593.
[68 ] Rohr J , Angew. Chem. Int. Ed. Engl. , 1995, 34 (8) , 881~ 885.
[69 ] Carell T , Wintner E A et al. , Chemistry &Biology , 1995, 2 (3) , 171~ 183.
[70 ] Carell T , Wintner E A , Bashir-Hashemi A , Rebek J Jr, Angew. Chem. Int. Ed. Engl. , 1994, 33(20) , 2059~ 2061.
[71 ] Carell T , Wintner E A , Rebek J Jr, Angew. Chem. Int. Ed. Engl. , 1994, 33 (20) , 2061~ 2064.
[72 ] Smith P W , Lai J Y Q , Whitington A R, Cox B, Houston J G, Stylli C H, Banks M N , Tiller P R,Biomed. Chem. Lett. , 1994, 4, 2821~ 2824.
[73 ] Pirrung M C, Chen J , J. Am. Chem. Soc. , 1995, 117, 1240~ 1245.
[74 ] Merrifield R B, J. Am. Chem. Soc. , 1963, 85, 2149~ 2154.
[75 ] Knapp D R, Oatis J E, Papac D I, Int. J. Peptide Protein Res. , 1993, 42, 259~ 263.
[76 ] Meldal M , Holm C B, Bojesen G, Jakobsen M H, Holm A , Int. J. Peptide Protein Res. , 1993, 41,250~ 260.
[77 ] DeWitt S H, Schroeder M C, Stankovic C J , Strode J E, Czarnik A W , Drug Development Research, 1994, 33, 116~ 124.
[78 ] Bartak Z, Bolf J , Kalousek J , Methods: A Companion to Methods in Enzymology , 1994, 6, 432~437.
[79 ] Geysen H M , Barteling R H, Meloen R H, Proc. Natl. Acad. Sci. USA , 1985, 82, 178~ 182.
80 ] Valerio R M , Bray A M , Campbell R A , Dipasquale A , Margellis C, Rodda S T , Geysen H M ,Maeji N J , Int. J. Peptide Protein Res. , 1993, 42, 1~ 9.
[81 ] Lebl M , Krchnak V , Safar P, Stierandova A , Sepetov N F, Kocis P, Lam K S, Techniquesin Protein Chemistry , 1994, 541.
[82 ] Tam J P, Proc. Natl. Acad. Sci. USA , 1988, 85, 5409~ 5413.
[83 ] 张所德, 刘刚, 夏叔泉, 军事医学科学院毒物药物研究所硕士研究论文, 1996, 6 月1
[84 ] Bunin B A , Ellman J A , J. Am. Chem. Soc. , 1992, 114, 10997~ 10998.
[85 ] Bunin B A , Plunkett M J , Ellman J A , Proc. Natl. Acad. Sci. USA , 1994, 6, 4708~ 4712.
[86 ] Ellman J A , Accountsof Chemical Research, 1996, 29 (3) , 132~ 143.
[87 ] Plunkett M J , Ellman J A , J. Am. Chem. Soc. , 1995, 117, 3306~ 3307.
[88 ] Dankwardt S M , Phan T M , Krstenansky J L , Molecular Diversity , 1996, 1, 1.
[89 ] DeWitt S H, Kiely J S, Stankovic C J et al. , Proc. Natl. Acad. Sci. USA , 1993, 90, 6909.
[90 ] Virgilio A A , Ellman J A , J. Am. Chem. Soc. , 1994, 116, 11580~ 11581.
[91 ] Chen C, RandallL A A , Miller B, JonesA D, Kurth M J , J. Am. Chem. Soc. , 1994, 116, 2661~2662.
[92 ] Cho C Y, Moran E J , Cherry S R, Stephans J C, Fordor S P A , Adams C L , Sundaram A , Jacobs J W , Schultz P G, Science, 1993, 261, 1303~ 1305.
[93 ] Moran E J , Wilson T E, Cho C Y, Biopolymers, 1995, 37, 213~ 219.
[94 ] Burgess K, Linthicum D S, Shin H W , Angew. Chem. Int. Ed. Engl. , 1995, 34, 907~ 909.
[95 ] Gennari C, Nestler H P, Salom B, Still W C, Angew. Chem. Int. Ed. Engl. , 1995, 34, 1763~1765.
[96 ] Gordon D W , Steele J , Biomed. Chem. Lett. , 1995, 5, 47~ 50.
[97 ] Halcomb R L , Huang H M , Wong C H, J. Am. Chem. Soc. , 1994, 116, 11315~ 11322.
[98 ] Roberge J Y, Beebe X, Danishefsky S J , Science, 1995, 269, 202~ 204.
[99 ] Yan L , Taylor C M , Goodnow R, Kahne D, J. Am. Chem. Soc. , 1994, 116, 6953~ 6954.
[100 ] Danishefsky S J , McClure K F, Randolph J T , Ruggeri R B, Science, 1993, 260, 1307~ 1309.
[101 ] Vetter D, Gallop M A , Bioconjugate Chemistry , 1995, 6, 316~ 318.
[102 ] Vetter D, Tate E M , Gallop M A , Bioconjugate Chemistry , 1995, 6, 319~ 322.
[103 ] Vetter D, Tumelty D, Singh S Q , Gallop M A , Angew. Chem. Int. Ed. Engl. , 1995, 34, 60~63.
[104 ] Goff D A , Zuckermann R N , J. Org. Chem. , 1995, 60, 5748~ 5749.
[105 ] Gordeev M F, Patel D V , Gordon E M , J. Org. Chem. , 1996, 61, 924~ 928.
[106 ] Meutermans W D F, Alowood P F, Tetrahedron Lett. , 1995, 36, 7709~ 7712.
[107 ] Murphy M M , Schullek J R, Gordon E M , Gallop M A , J. Am. Chem. Soc. , 1995, 117, 7029~7030.
[108 ] Patek M , Brake B, Lebl M , Tetrahedron Lett. , 1995, 36, 2227~ 2230.
[109 ] Holmes C P, Chinn J P, Look G C, J. Org. Chem. , 1995, 60, 7328~ 7333.
[110 ] Boojamara C G, Burow K M , Ellman J A , J. Org. Chem. , 1995, 60, 5742~ 5743.
[111 ] Goff D A , Zuckermann R N , J. Org. Chem. , 1995, 60, 5744~ 5745.
[112 ] Kassarjian A , Schellenberger V , Turck C W , Peptide Res. , 1993, 6, 129~ 133.
[113 ] Needels M C, JonesD G, Tate E H, Heinkel G L , Kochersperger L M , Dower W J , Barrett R W ,Gallop M A , Proc. Natl. Acad. Sci. USA , 1993, 90, 10700~ 10704.
[114 ] Nielsen J , Brenner R A , Janda K D, J. Am. Chem. Soc. , 1993, 115, 9812~ 9813.
[115 ] Ohlmeyer M H, Swanson R N , Dillard L W , Reader J C, Asouline G, Kobayashi R, Wigler M ,Still W C, Proc. Natl. Acad. Sci. USA , 1993, 90, 10922~ 10926.
[116 ] Smith M H, Lam K S, Hersh E M , Lebl M , Grimes W J , Mol. Immunol. , 1994, 31, 1431~ 1437.
[117 ] Salmon S E, Lam K S, Lebl M , Kandola A , Khattri P S, Wade S, Pátek M , Kocis P, Krchnák V ,Thorpe D, Felders S, Proc. Natl. Acad. Sci. USA , 1993, 90, 11708~ 11712.
[118 ] Lam A S, Lebl M , Immunomethods 1, 1992, 11~ 15.
[119 ] Wu J Z, Ma Q N , Lam K S, Biochemistry , 1994, 33, 14825~ 14833.
[120 ] Lam K S, Wu J Z, Lou Q , Int. J. Peptide Protein Res. , 1995, 45, 587~ 592.
[121 ] Lam K S, Zhao Z G, Wade S, Krchnak V , Lebl M , Drug Development Research, 1994, 33, 157~160.
[122 ] Lam K S, Lebl M , Methods: A Companion to Methods in Enzymology , 1994, 6, 372~ 380.
[123 ] Lam K S, Wade S, Abdul-Latif F, Lebl M , J. Immunological Methods, 1995, 180, 219~ 223.
[124 ] Lebl M , Patek M , Kocis P, Krchnak V , Hruby V J , Salmon S E, Lam K S, Int. J. Peptide Protein Res. , 1993, 41, 201~ 203.
[125 ] Richter L S, Spellmeyer D V , Martin E J , Figliozzi G M , Zuckermann R N ,in Combinatorial Peptide and Nonpeptide Libraries (ed. Jung G) , VCH, 1996, 389. |