[1] Dawson P E, Muir T W, Lewis L C, Kent S B H. Science, 1994, 266: 776.
[2] Durek T, Torbeev V Y, Kent S B H. Proc. Natl. Acad. Sci. U. S. A., 2007, 104: 4846.
[3] Torbeev V Y, Kent S B H. Angew. Chem. Int. Ed., 2007, 46: 1667.
[4] McGinty R K, Kim J, Chatterjee C, Roeder R G, Muir T W. Nature, 2008, 453: 812.
[5] Fang G M, Wang J X, Liu L. Angew. Chem. Int. Ed., 2012, 51: 10347.
[6] Fang G M, Li Y M, Shen F, Huang Y C, Li J B, Lin Y, Cui H C, Liu L. Angew. Chem. Int. Ed., 2011, 50: 7645.
[7] Zheng J S, Chang H N, Wang F L, Liu L. J. Am. Chem. Soc., 2011, 133: 11080.
[8] Zheng J S, Huang Y C, Tang S, Liu L. Acc. Chem. Res., 2013, 46: 2475.
[9] Zheng J S, Tang S, Qi J Q, Wang Z P, Liu L. Nat. Protoc., 2013, 8: 2483.
[10] Chen Y X, Koch S, Uhlenbrock K, Weise K, Das D, Gremer L, Brunsveld L, Wittinghofer A, Winter R, Triola G, Waldmann H. Angew. Chem. Int. Ed., 2010, 49: 6090.
[11] Huang Y C, Li Y M, Chen Y, Pan M, Li Y T, Yu L, Guo Q X, Liu L. Angew. Chem. Int. Ed., 2013, 52: 4858.
[12] Dawson P E, Kent S B H. Biochem., 2000, 69: 923.
[13] Malins L R, Cergol K M, Payne R G. ChemBioChem, 2013, 14: 559.
[14] Dumas A, Spicer C D, Gao Z H, Takehana T, Lin Y A, Yasukohchi T, Davis B G. Angew. Chem. Int. Ed., 2013, 52: 3916.
[15] Binschik J, Mootz H D. Angew. Chem. Int. Ed., 2013, 52: 4260.
[16] Adams A L, Macmillan D. J. Pept. Sci., 2013, 19: 65.
[17] Fang G M, Cui H K, Zheng J S, Liu L. ChemBioChem, 2010, 11: 1061.
[18] Zheng J S, Cui H K, Fang G M, Xi W X, Liu L. ChemBioChem, 2010, 11: 511.
[19] Spokoyny A M, Zou Y K, Ling J J, Yu H T, Lin Y S, Pentelute B L. J. Am. Chem. Soc., 2013, 135: 5946.
[20] Gordon W R, Bang D, Hoff W D, Kent S B H. Bioorg. Med. Chem., 2013, 21: 3436.
[21] Li Y M, Yang M Y, Huang Y C, Li Y T, Chen P R, Liu L. ACS Chem. Biol., 2012, 7: 1015.
[22] Cronican J J, Thompson D B, Beier K T, McNaughton B R, Cepko C L, Liu D R. ACS Chem. Biol., 2010, 5: 747.
[23] Lawrence M S, Phillips K J, Liu D R. J. Am. Chem. Soc., 2007, 129: 10110.
[24] McNaughton B R, Cronican J J, Thompson D B, Liu D R. Proc. Natl. Acad. Sci. U. S. A., 2009, 106: 6111.
[25] Jenssen H, Aspmo S I. Methods Mol. Biol., 2008, 494: 177.
[26] Schafmeister C E, Po J, Verdine G L. J. Am. Chem. Soc., 2000, 122, 5891.
[27] Blackwell H E, Grubbs R H. Angew. Chem. Int. Ed., 1998, 37: 3281.
[28] Dastlik K A, Sundermerier U, Johns D M, Chen Y, Williams R M. Synlett, 2005, 4: 693.
[29] Williams R M, Im M N. J. Am. Chem. Soc., 1991, 113: 9276.
[30] Kim Y W, Grossmann T N, Verdine G L. Nat. Protoc., 2011, 6: 761.
[31] Muppidi A, Li X L, Chen J D, Lin Q. Bioorg. Med. Chem. Lett., 2011, 21: 7412.
[32] Greenfield N, Fasman G D. Biochem, 1969, 8: 4108.
[33] Baek S, Kutchukian P S, Verdine G L, Huber R, Holak T A, Lee K W, Popowicz G M. J. Am. Chem. Soc., 2012, 134: 103.
[34] Phillips C, Roberts L R, Schade M, Bazin R, Bent A, Davies N L, Moore R, Pannifer A D, Pickford A R, Prior S H, Read C M, Scott A, Brown D G, Xu B, Irving S L. J. Am. Chem. Soc., 2011, 133: 9696.
[35] Bernal F, Tyler A F, Korsmeyer S J, Walensky L D, Verdine G L. J. Am. Chem. Soc., 2007, 129: 2456.
[36] Moellering R E, Cornejo M, Davis T N, Bianco C D, Aster J C, Blacklow S C, Kung A L, Gilliland D G, Verdine G L, Bradner J E. Nature, 2009, 462: 182.
[37] Walensky L D, Kung A L, Escher I, Malia T J, Barbuto S, Wright R D, Wagner G, Verdine G L, Korsmeyer S J. Science, 2004, 305: 1466.
[38] Zhang H, Zhao Q, Bhattacharya S, Waheed A A, Tong X, Hong A, Heck S, Curreli F, Goger M, Cowburn D, Freed E O, Debnath A K. J. Mol. Biol., 2008, 378: 565.
[39] Bautista A D, Appelbaum J S, Craig C J, Michel J, Schepartz A. J. Am. Chem. Soc., 2010, 132: 2904.
[40] Bird G H, Bernal F, Pitter K, Walensky L D. Methods Enzymol., 2008, 446: 369.
[41] Verdine G L, Hilinski G J. Methods in Enzymology, 2012, 503: 3.
[42] Gavathiotis E, Suzuki M, Davis M L, Pitter K, Bird G H, Katz S G, Tu H C, Kim H, Cheng E H, Tjandra N T, Walens L D. Nature, 2008, 455: 1076.
[43] Pitter K, Bernal F, Labelle J, Walensky L D. Methods Enzymol., 2008, 446: 387.
[44] Stewart M L, Fire E, Keating A E, Walensky L D. Nat. Chem. Biol., 2010, 6: 595.
[45] Walensky L D, Pitter K, Morash J, Oh K J, Barbuto S, Fisher J, Smith E, Verdine G L, Korsmeyer S J. Mol. Cell, 2006, 24: 199.
[46] Bernal F, Wade M, Godes M, Davis T N, Whitehead D G, Kung A L, Wahl G M, Walensky L D. Cancer Cell, 2010, 18: 411.
[47] Danial N N, Gramm C F, Scorrano L, Zhang C-Y, Krauss S, Ranger A M, Datta S R, Greenberg M E, Licklider L J, Lowell B B, Gygi S P, Korsmeyer S J. Nature, 2003, 424: 952.
[48] Plas D R, Thompson C B. Trends Endocrin. Met., 2002, 13: 74.
[49] Pinton P, Rizzuto R. Cell Death Differ., 2006, 13: 1409.
[50] Karbowski M, Norris K L, Cleland M M, Jeong S Y, Youle R J. Nature, 2006, 443: 658.
[51] Sticht J, Humbert M, Findlow S, Bodem J, Muller B, Dietrich U, Werner J, Krausslich H G. Nat. Struct. Mol. Biol., 2005, 12: 671.
[52] Sakalian M, McMurtrey C P, Deeg F J, Maloy C W, Li F, Wild C T, Salzwedel K. J. Virol., 2006, 80: 5715.
[53] Bird G H, Madani N, Perry A F, Princiotto A M, Supko J G, He X Y, Gavathiotis E, Sodroski J G, Walensky L D. Proc. Natl. Acad. Sci. U. S. A., 2010, 107: 14093.
[54] Cui H K, Zhao B, Li Y H, Guo Y, Hu H, Liu L, Chen Y G. Cell Res., 2013, 23: 581.
[55] Cui H K, Qing J, Guo Y, Wang Y J, Cui L J, He T H, Zhang L Q, Liu L. Bioorg. Med. Chem., 2013, 21: 3547.
[56] Cascales L, Craik D J. Org. Biomol. Chem., 2010, 8: 5035.
[57] Göransson U, Burman R, Gunasekera S, Strömstedt A A, Rosengren K J. J. Biol. Chem., 2012, 287: 27001.
[58] Zheng J S, Tang S, Guo Y, Chang H N, Liu L. ChemBioChem, 2012, 13: 542.
[59] Cowper B, Craik D J, Macmillan D. ChemBioChem 2013, 14: 809.
[60] Zheng J S, Chang H N, Shi J, Liu L. Sci. China Chem., 2012, 55: 64.
[61] Thorstholm L, Craik D J. Drug Discov. Today Tech. 2012, 9: e13.
[62] Daly N L, Rosengren K J, Craik D J. Curr. Protein Pept. Sci., 2004, 5: 297.
[63] Göransson U, Svangård E, Claeson P, Bohlin L. Curr. Protein Pept. Sci., 2004, 5: 317.
[64] Tang Y Q, Yuan J, Osapay G, Osapay K, Tran D, Miller C J, Ouellette A J, Selsted M E. Science, 1999, 286: 498.
[65] Cui H K, Guo Y, He Y, Wang F L, Chang H N, Wang Y J, Wu F M, Tian C L, Liu L. Angew. Chem. Int. Ed., 2013, 52: 9558. |